Jiajie Zhang

Dr. Jiajie Zhang

School of Pharmaceutical Science, Southern Medical University, Guangzhou, Guangdong, China

Research Focus & Metrics

Academic Career Length

23Years (2004-Present)

(Calculated once Scilit publication data is synced: current year − year of first publication + 1)

Representative Publications

View All Publications
5 January 2009 in Acta Pharmacologica Sinica
Verified
Journal Article
Closed access
SWShao-Yu Wu
Shao-Yu Wu
GWGuang-Fa Wang
Guang-Fa Wang
ZLZhong-Qiu Liu
Zhong-Qiu Liu
JRJin-Jun Rao
Jin-Jun Rao
LLLin Lü
Lin Lü
JZJiajie Zhang
Jiajie Zhang

15 November 2011 in Inflammation
Verified
Journal Article
Closed access
PDF file
PYPeng-Jiu Yu
Peng-Jiu Yu
HJHong Jin
Hong Jin
JZJun-Yan Zhang
Jun-Yan Zhang
GWGuang-Fa Wang
Guang-Fa Wang
JLJing-Rong Li
Jing-Rong Li
SWShu-Guang Wu
Shu-Guang Wu

6 April 2009 in Acta Pharmacologica Sinica
Verified
Journal Article
Closed access
GWGuang-Fa Wang
Guang-Fa Wang
SWShao-Yu Wu
Shao-Yu Wu
JRJin-Jun Rao
Jin-Jun Rao
LLLin Lü
Lin Lü
WXWei Xu
Wei Xu
JZJiajie Zhang
Jiajie Zhang

1 August 2016 in European Journal of Medicinal Chemistry
Verified
Journal Article
Closed access
JHJu Hou
Ju Hou
SWShanhe Wan
Shanhe Wan
GWGuangfa Wang
Guangfa Wang
TZTingting Zhang
Tingting Zhang
ZLZhonghuang Li
Zhonghuang Li
JZJiajie Zhang
Jiajie Zhang

1 July 2018 in European Journal of Medicinal Chemistry
Verified
Journal Article
Closed access
YWYuanyuan Wang
Yuanyuan Wang
SWShanhe Wan
Shanhe Wan
ZLZhonghuang Li
Zhonghuang Li
YFYu Fu
Yu Fu
GWGuangfa Wang
Guangfa Wang
XWXiaoyun Wu
Xiaoyun Wu

16 July 2013 in ACS Medicinal Chemistry Letters
Verified
Journal Article
Open access
JLJingrong Li
Jingrong Li
NWNan Wu
Nan Wu
TYTian Yuanxin
Tian Yuanxin
JZJiajie Zhang
Jiajie Zhang
SWShuguang Wu
Shuguang Wu
A series of novel aminopyridyl/pyrazinyl-substituted spiro[indoline-3,4′-piperidine]-2-ones were designed, synthesized, and tested in various in vitro/in vivo pharmacological and antitumor assays. 6-[6-Amino-5-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-pyridyl]-1′-methylspiro[indoline-3,4′-piperidine]-2-one (compound 5b or SMU-B) was identified as a potent, highly selective, well-tolerated, and orally efficacious c-Met/ALK dual inhibitor, which showed pharmacodynamics effect by inhibiting c-Met phosphorylation in vivo and significant tumor growth inhibitions (>50%) in GTL-16 human gastric carcinoma xenograft models.