The present article reviews the most important developing strategies in light-induced nanomedicine, based on the combination of porphyrinoid photosensitizers with a wide variety of biomolecules and biomolecular assemblies.

Novel zinc phthalocyanine (ZnPc)/fullerene ligand (L) ensembles are assembled following simple biomimetic principles, which upon photoexcitation give rise to intra complex electron transfer quenching of the ¹*ZnPc fluorescence.